A mixture of alkaloids with diverse biological activities; blocks norepinephrine-induced reflex vasodilation and vasoconstriction in dogs when injected into the kidney at a dose of 0.15 mg; blocks norepinephrine-induced cAMP production in rat brain cortical homogenates ex vivo in a dose-dependent manner; acts as an erectogenic agent in rats

Ergoloid (mesylates) – 100 mg

Brand:
Cayman
CAS:
8067-24-1
Storage:
-20
UN-No:
Non-Hazardous - /

Ergoloid is a mixture of the ergot alkaloids dihydroergocornine, dihydroergocrystine, and dihydroergocryptine.{37285} It blocks reflex vasodilation and vasoconstriction induced by norepinephrine (Item No. 16673) in dogs when injected into the kidney at a dose of 0.15 mg. Ergoloid blocks norepinephrine-induced cAMP production in rat brain cortical homogenates ex vivo in a dose-dependent manner.{37286} It also acts as an erectogenic agent in rats.{37287} Formulations containing ergoloid have been used in the treatment of migraine headaches and vascular dementias.  

 

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SKU: 24095 - 100 mg Category:

Description

A mixture of alkaloids with diverse biological activities; blocks norepinephrine-induced reflex vasodilation and vasoconstriction in dogs when injected into the kidney at a dose of 0.15 mg; blocks norepinephrine-induced cAMP production in rat brain cortical homogenates ex vivo in a dose-dependent manner; acts as an erectogenic agent in rats

Formal name: dihydro-ergotoxine, monomethanesulfonate

Synonyms: 

Molecular weight: 2,715.30

CAS: 8067-24-1

Purity: ≥95%

Formulation: A solid

Product Type|Biochemicals|Natural Products|Alkaloids||Product Type|Biochemicals|Natural Products|Microbial Metabolites||Research Area|Cardiovascular System|Cardiovascular Diseases||Research Area|Cardiovascular System|Vasculature|Vasoconstriction||Research Area|Cardiovascular System|Vasculature|Vasodilation||Research Area|Neuroscience|Pain Research

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