A fatty acid amide; inhibits rat mEH (Ki = 70 nM); inhibits porcine pancreatic and human synovial PLA2; induces physiological sleep in rats at 10 mg/animal

Elaidamide – 10 mg

Brand:
Cayman
CAS:
4303-70-2
Storage:
-20
UN-No:
Non-Hazardous - /

Elaidamide is a fatty acid amide that has been found in the cerebrospinal fluid of sleep-deprived cats.{1317} It inhibits rat microsomal epoxide hydrolase (mEH; Ki = 70 nM).{50370} Elaidamide also inhibits porcine pancreatic and human synovial phospholipase A2 (PLA2).{50371} In vivo, elaidamide (10 mg/animal) induces physiological sleep in rats.{1317}  

 

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Description

A fatty acid amide; inhibits rat mEH (Ki = 70 nM); inhibits porcine pancreatic and human synovial PLA2; induces physiological sleep in rats at 10 mg/animal

Formal name: 9E-octadecenamide

Synonyms:  (E)-9,10-Octadecenamide|Elaidic Acid amide

Molecular weight: 281.5

CAS: 4303-70-2

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Lipids|Fatty Amides||Product Type|Biochemicals|Small Molecule Inhibitors|Phospholipases||Product Type|Biochemicals|Small Molecule Inhibitors|Prolyl Hydroxylation Enzymes||Research Area|Neuroscience|Behavioral Neuroscience|Sleep & Biological Rhythms

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