An NMDA receptor antagonist; selectively inhibits glutamate-induced currents in Xenopus oocytes expressing rat NR2C and NR2D subunit-containing NMDA receptors (IC50s = 8.5 and 2.7 µM

DQP1105 – 10 mg

Brand:
Cayman
CAS:
380560-89-4
Storage:
-20
UN-No:
Non-Hazardous - /

DQP1105 is an NMDA receptor antagonist.{52769} It selectively inhibits glutamate-induced currents in Xenopus oocytes expressing rat NR2C and NR2D subunit-containing NMDA receptors (IC50s = 8.5 and 2.7 µM, respectively) over NR2A, NR2B, NRA1, and NRK2 subunit-containing receptors (IC50s = 206, 121, 198, and 153 µM, respectively).  

 

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SKU: 31121 - 10 mg Category:

Description

An NMDA receptor antagonist; selectively inhibits glutamate-induced currents in Xenopus oocytes expressing rat NR2C and NR2D subunit-containing NMDA receptors (IC50s = 8.5 and 2.7 µM, respectively) over NR2A, NR2B, NRA1, and NRK2 subunit-containing receptors (IC50s = 206, 121, 198, and 153 µM, respectively)

Formal name: 5-(4-bromophenyl)-3-(1,2-dihydro-6-methyl-2-oxo-4-phenyl-3-quinolinyl)-4,5-dihydro-γ-oxo-1H-pyrazole-1-butanoic acid

Synonyms: 

Molecular weight: 558.4

CAS: 380560-89-4

Purity: ≥98%

Formulation: A solid

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