An active metabolite of donepezil; inhibits ChE activity in human erythrocytes in a concentration-dependent manner

Donepezil N-oxide – 500 µg

Brand:
Cayman
CAS:
120013-84-5
Storage:
-20
UN-No:
Non-Hazardous - /

Donepezil N-oxide is an active metabolite of the acetylcholinesterase inhibitor donepezil (Item No. 13245).{47251} Donepezil N-oxide inhibits cholinesterase (ChE) activity in human erythrocytes in a concentration-dependent manner, exhibiting 45.5% inhibition when used at a concentration of 20 µM.{47252}  

 

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SKU: 27174 - 500 µg Category:

Description

An active metabolite of donepezil; inhibits ChE activity in human erythrocytes in a concentration-dependent manner

Formal name: 2,3-dihydro-5,6-dimethoxy-2-[[1-oxido-1-(phenylmethyl)-4-piperidinyl]methyl]-1H-inden-1-one

Synonyms: 

Molecular weight: 395.5

CAS: 120013-84-5

Purity: ≥98%

Formulation: A solid

Product Type|Biochemicals|Small Molecule Inhibitors|Acetylcholine Turnover||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Neuroscience|Behavioral Neuroscience|Learning & Memory||Research Area|Neuroscience|Neurodegenerative Disorders|Alzheimer’s Disease

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