A local anesthetic that

Dimethocaine (hydrochloride) – 5 mg

Brand:
Cayman
CAS:
553-63-9
Storage:
-20
UN-No:
Non-Hazardous - /

Dimethocaine is a local anesthetic that, because of its similarity in action to cocaine, has potential for abuse. This compound completely inhibits dopamine uptake in rat striatal synaptosomes with an IC50 value of 1.2 µM comparable to that of cocaine (IC50 = 0.7 µM).{24176} As a result, dimethocaine dose-dependently substitutes for cocaine in drug discrimination tests in rats and rhesus monkeys.{24175,23694} This product is intended for forensic and research purposes.  

 

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SKU: 11159 - 5 mg Category:

Description

A local anesthetic that, because of its similarity in action to cocaine, has potential for abuse; completely inhibits dopamine uptake in rat striatal synaptosomes with an IC50 value (1.2 µM) comparable to that of cocaine (IC50 = 0.7 µM); substitutes for cocaine in drug discrimination tests in rats and rhesus monkeys

Formal name: 3-(diethylamino)-2,2-dimethyl-1-(4-aminobenzoate)-1-propanol, monohydrochloride

Synonyms: 

Molecular weight: 314.9

CAS: 553-63-9

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Sedatives & Muscle Relaxers

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