An oxazolidinone antibiotic; is active against a wide range of Gram-positive bacterial clinical isolates (MICs = 0.125-4 μg/ml); increases survival in mouse models of systemic MRSA

Delpazolid – 25 mg

Brand:
Cayman
CAS:
1219707-39-7
Storage:
-20
UN-No:
Non-Hazardous - /

Delpazolid is an oxazolidinone antibiotic.{48191} It is active against a wide range of Gram-positive bacterial clinical isolates, including resistant strains of several species, such as methicillin-resistant S. aureus (MRSA), methicillin-resistant coagulase-negative staphylococci (MRCNS), and penicillin-resistant S. pneumoniae (MICs = 0.125-4 μg/ml). Delpazolid increases survival in mouse models of systemic MRSA, E. faecalis, S. pneumoniae, and H. influenzae infection (ED50s = 2.96, 4.53, 2.28, and 9.96 mg/kg, respectively).  

 

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SKU: 25532 - 25 mg Category:

Description

An oxazolidinone antibiotic; is active against a wide range of Gram-positive bacterial clinical isolates (MICs = 0.125-4 μg/ml); increases survival in mouse models of systemic MRSA, E. faecalis, S. pneumoniae, and H. influenzae infection (ED50s = 2.96, 4.53, 2.28, and 9.96 mg/kg, respectively)

Formal name: (5R)-3-[4-(5,6-dihydro-1-methyl-1,2,4-triazin-4(1H)-yl)-3-fluorophenyl]-5-(hydroxymethyl)-2-oxazolidinone

Synonyms:  LCB01-0371

Molecular weight: 308.3

CAS: 1219707-39-7

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Antibiotics|Oxazolidinones||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Bacterial Diseases|MRSA||Research Area|Infectious Disease|Bacterial Diseases|Pneumonia

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