A muscarinic receptor antagonist (Kis = 1.62

Cyclopentolate (hydrochloride) – 10 mg

Brand:
Cayman
CAS:
5870-29-1
Storage:
-20
UN-No:
Non-Hazardous - /

Cyclopentolate is an antagonist of muscarinic acetylcholine receptors (Kis = 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively).{27107} It inhibits carbachol-induced contraction of isolated human iris sphincter, circular ciliary muscle, and longitudinal ciliary muscle (Kbs = 7.9, 15.8, and 12.5 nM, respectively).{41287} Formulations containing cyclopentolate have been used to induce pupil dilation and to prevent the eye from accommodating for near vision.  

 

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SKU: 23944 - 10 mg Category:

Description

A muscarinic receptor antagonist (Kis = 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively); inhibits carbachol-induced contraction of isolated human iris sphincter, circular ciliary muscle, and longitudinal ciliary muscle (Kbs = 7.9, 15.8, and 12.5 nM, respectively)

Formal name: α-(1-hydroxycyclopentyl)–benzeneacetic acid, 2-(dimethylamino)ethyl ester, monohydrochloride

Synonyms:  (±)-Cyclopentolate

Molecular weight: 327.9

CAS: 5870-29-1

Purity: ≥98%

Formulation: A solid

Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Neuroscience|Ophthalmology

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