A corticosteroid that potently activates the glucocorticoid receptor (IC50 = 3 nM)

Clobetasol Propionate – 500 mg

Brand:
Cayman
CAS:
25122-46-7
Storage:
-20
UN-No:
Non-Hazardous - /

Clobetasol propionate is a corticosteroid that potently activates the glucocorticoid receptor (IC50 = 3 nM).{33297} Formulations containing clobetasol propionate are used topically to suppress inflammatory skin conditions.{33296,33298}  

 

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Description

A corticosteroid that potently activates the glucocorticoid receptor (IC50 = 3 nM)

Formal name: 21-chloro-9-fluoro-11β-hydroxy-16β-methyl-17-(1-oxopropoxy)-pregna-1,4-diene-3,20-dione

Synonyms:  CCl-4725|CGP 9555|Clobetasol 17-Propionate

Molecular weight: 467

CAS: 25122-46-7

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Glucocorticoids & Mineralocorticoids||Research Area|Immunology & Inflammation

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