A sympathomimetic β2-adrenoceptor agonist that relaxes bronchial smooth muscle and at higher doses acts as an anabolic steroid

Clenbuterol (hydrochloride) – 25 mg

Brand:
Cayman
CAS:
21898-19-1
Storage:
-20
UN-No:
De Minimis - 2811 / 6.1

Clenbuterol is a sympathomimetic β2-adrenoceptor agonist that has been used as a bronchodilator (20 μg per dose in humans) in the treatment of pulmonary diseases such as asthma.{23878,23874} At higher doses (2 mg/kg/day in rats), clenbuterol acts as an anabolic steroid, favoring skeletal muscle protein synthesis at the expense of fat deposition.{23875} Because of this property, clenbuterol has been illegally used by athletes to enhance performance, by dieters to encourage weight loss, and by livestock farmers to produce animals with leaner meat.{23876,23880} The use of clenbuterol is banned by the U.S. Food and Drug Administration as well as the International Olympic Committee and is prohibited for use in food-producing animals in the U.S., the European Union, and China.{5878} Clenbuterol can also produce relaxation of smooth muscle in the uterus and has been used in the short-term postponement of parturition in veterinary obstetrical procedures.{23877}  

 

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Description

A sympathomimetic β2-adrenoceptor agonist that relaxes bronchial smooth muscle and at higher doses acts as an anabolic steroid, promoting skeletal muscle protein synthesis

Formal name: 4-amino-3,5-dichloro-α-[[(1,1-dimethylethyl)amino]methyl]-benzenemethanol, monohydrochloride

Synonyms:  NAB 365

Molecular weight: 313.7

CAS: 21898-19-1

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Endocrinology & Metabolism|Hormones & Receptors||Research Area|Endocrinology & Metabolism|Reproductive Biology||Research Area|Immunology & Inflammation|Pulmonary Diseases|Asthma

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