A synthetic progestin; binds to progesterone

Chlormadinone Acetate – 250 mg

Brand:
Cayman
CAS:
302-22-7
Storage:
-20
UN-No:
Non-Hazardous - /

Chlormadinone acetate is a synthetic progestin.{45702} It binds to progesterone, androgen, and glucocorticoid receptors in vitro (Kis = 2.5, 3.8, and 16 nM, respectively, for the human receptors). Chlormadinone acetate increases the number of endometrial glands and uterine weight in β-estradiol-primed rabbits when administered at a dose of 45 µg/kg per day for five days. Chlormadinone acetate reduces testosterone-induced increases in the seminal vesicle weight of castrated male rats when administered at doses of 4.6 and 21.5 mg/kg per day for eight days.  

 

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SKU: 29392 - 250 mg Category:

Description

A synthetic progestin; binds to progesterone, androgen, and glucocorticoid receptors in vitro (Kis = 2.5, 3.8, and 16 nM, respectively, for the human receptors); increases the number of endometrial glands and uterine weight in β-estradiol-primed rabbits at 45 µg/kg per day for five days; reduces testosterone-induced increases in the seminal vesicle weight of castrated male rats at 4.6 and 21.5 mg/kg per day for eight days

Formal name: 17-(acetyloxy)-6-chloro-pregna-4,6-diene-3,20-dione

Synonyms:  NSC 92338

Molecular weight: 404.9

CAS: 302-22-7

Purity: ≥98%

Formulation: A solid

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