A stable analog of Δ9-THC; exhibits high affinity for the CB1 and CB2 receptors with Ki values of 5.2 and 13 nM

CB-25 – 5 mg

Brand:
Cayman
CAS:
869376-63-6
Storage:
-20
UN-No:
Non-Hazardous - /

CB-25 is a stable analog of Δ9-tetrahydrocannabinol (THC) and anandamide (AEA). It exhibits high affinity for the central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors with Ki values of 5.2 and 13 nM, respectively. CB-25 behaves as an inverse agonist for the CB1 receptor as assessed in a cyclic AMP (cAMP) functional assay.{14815,14816}  

 

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SKU: 10010116 - 5 mg Category:

Description

A stable analog of Δ9-THC; exhibits high affinity for the CB1 and CB2 receptors with Ki values of 5.2 and 13 nM, respectively, also it behaves as an inverse agonist for the CB1 receptor as assessed in a cyclic AMP functional assay

Formal name: N-cyclopropyl-11-(3-hydroxy-5-pentylphenoxy)-undecanamide

Synonyms: 

Molecular weight: 403.6

CAS: 869376-63-6

Purity: ≥98%

Formulation: A crystalline solid

Application||Product Type|Biochemicals|Receptor Pharmacology|Inverse Agonists||Research Area|Neuroscience|Cannabinoid Research|CB1 & CB2 Receptors

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