A cell-active analog of the lysine acetyltransferase inhibitor CPTH2 (Item No. 12086) that contains an alkyne moiety for use in click chemistry reactions; used to study changes in nuclear architecture associated with cancer and certain laminopathies

CAY10685 – 5 mg

Brand:
Cayman
CAS:
1613116-16-7
Storage:
-20
UN-No:
Non-Hazardous - /

CAY10685 is a cell-active analog of the lysine acetyltransferase inhibitor CPTH2 (Item No. 12086) that contains an alkyne moiety for use in click chemistry reactions.{26026} Its ability to inhibit N-acetyltransferase 10 activity has been used to modulate chromatin organization in order to study changes in nuclear architecture associated with cancer and certain laminopathies.{26026}  

 

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Description

A cell-active analog of the lysine acetyltransferase inhibitor CPTH2 (Item No. 12086) that contains an alkyne moiety for use in click chemistry reactions; used to study changes in nuclear architecture associated with cancer and certain laminopathies

Formal name: 4-(4-chlorophenyl)-2-(2-cyclopentylidene-1-(prop-2-yn-1-yl)hydrazinyl)thiazole

Synonyms:  Click Tag™ CAY10685

Molecular weight: 329.8

CAS: 1613116-16-7

Purity: ≥98%

Formulation: A crystalline solid

Application|Click Chemistry||Product Type|Biochemicals|Labeling & Detection|Reactive Probes||Product Type|Biochemicals|Small Molecule Inhibitors|Acyltransferases||Research Area|Epigenetics, Transcription, & Translation|Writers|Histone Acetylation

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