Derivative of PGF1α containing an acetylenic fluorobenzene substituent in the lower side chain; binds to the recombinant human FP receptor with an IC50 value of about 0.5 µM

CAY10510 – 100 µg

Brand:
Cayman
CAS:
291303-34-9
Storage:
-20
UN-No:
De Minimis - 1173 / 3

The actions of many clinical prostaglandins, including those used for estrous synchronization and for reduction of intraocular pressure, are mediated through the FP receptor.{2959} CAY10510 is an analog of PGF2α containing an acetylenic fluorobenzene substituent in the lower side chain. CAY10510 has an IC50 of 0.5 µM when tested for binding to the recombinant human FP receptor.{14404}  

 

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SKU: 10009168 - 100 µg Category:

Description

Derivative of PGF1α containing an acetylenic fluorobenzene substituent in the lower side chain; binds to the recombinant human FP receptor with an IC50 value of about 0.5 µM

Formal name: 9α,11α,15-trihydroxy-17-fluorophenyl-18,19,20-trinor-prost-16-yn-1-oic acid, methyl ester

Synonyms: 

Molecular weight: 420.5

CAS: 291303-34-9

Purity: ≥98%

Formulation: A solution in ethyl acetate

Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway

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