A reversible caspase-3 inhibitor (IC50 = 23 nM); displays anti-apoptotic activity in Jurkat T cells treated with staurosporine

Caspase-3 Inhibitor VII – 5 mg

Brand:
Cayman
CAS:
745046-84-8
Storage:
-20
UN-No:
Non-Hazardous - /

Caspase-3 inhibitor VII is a 4-methylated pyrroloquinoline that reversibly inhibits caspase-3 (IC50 = 23 nM).{34501} It displays anti-apoptotic activity in Jurkat T cells treated with staurosporine (Item No. 81590).{34501}  

 

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Description

A reversible caspase-3 inhibitor (IC50 = 23 nM); displays anti-apoptotic activity in Jurkat T cells treated with staurosporine,

Formal name: 2-[2-(acetyloxy)ethyl]-4-methyl-8-(4-morpholinylsulfonyl)-1H-pyrrolo[3,4-c]quinoline-1,3(2H)-dione

Synonyms:  Ivachtin

Molecular weight: 447.5

CAS: 745046-84-8

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Caspases||Research Area|Cancer|Cell Death|Apoptosis||Research Area|Cell Biology|Cell Death|Apoptosis||Research Area|Cell Biology|Proteolysis|Cytosolic & Secreted Proteases

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