A histamine H3 receptor antagonist and histamine H1 receptor agonist; dilates pre-capillary arterioles and increases blood flow to the stria vascularis in guinea pigs; reduces olanzapine-induced weight gain and increased feeding behavior in female rats at 8 mg/kg

Betahistine (hydrochloride) – 1 g

Brand:
Cayman
CAS:
5579-84-0
Storage:
-20
UN-No:
Non-Hazardous - /

Betahistine is a histamine H3 receptor antagonist and histamine H1 receptor agonist.{45328} In vivo, betahistine dilates pre-capillary arterioles and increases blood flow to the stria vascularis in guinea pigs.{45329,45330} Betahistine (8 mg/kg) reduces weight gain and increased feeding behavior induced by olanzapine (Item No. 11937) in female rats.{45331} Formulations containing betahistine have been used in the treatment of balance disorders and vertigo symptoms associated with Meniere’s disease.  

 

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SKU: 27602 - 1 g Category:

Description

A histamine H3 receptor antagonist and histamine H1 receptor agonist; dilates pre-capillary arterioles and increases blood flow to the stria vascularis in guinea pigs; reduces olanzapine-induced weight gain and increased feeding behavior in female rats at 8 mg/kg

Formal name: N-methyl-2-pyridineethanamine, dihydrochloride

Synonyms: 

Molecular weight: 209.1

CAS: 5579-84-0

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology|Agonists||Product Type|Biochemicals|Receptor Pharmacology|Antagonists||Research Area|Endocrinology & Metabolism|Metabolic Diseases|Obesity||Research Area|Neuroscience

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