An internal standard for the quantification of apixaban by GC- or LC-MS

Apixaban-13C-d3 – 500 µg

Brand:
Cayman
CAS:
1261393-15-0
Storage:
-20
UN-No:
Non-Hazardous - /

Apixaban-13C-d3 is intended for use as an internal standard for the quantification of apixaban (Item No. 15427) by GC- or LC-MS. Apixaban is an orally bioavailable, selective inhibitor of both free and prothrombinase-bound factor Xa (Kis = 0.8 nM).{25094} In vivo, apixaban has antithrombotic effects in a rabbit model of venous thrombosis.  

 

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SKU: 25034 - 500 µg Category:

Description

An internal standard for the quantification of apixaban by GC- or LC-MS

Formal name: 4,5,6,7-tetrahydro-1-[4-(methoxy-13C-d3)phenyl]-7-oxo-6-[4-(2-oxo-1-piperidinyl)phenyl]-1H-pyrazolo[3,4-c]pyridine-3-carboxamide

Synonyms: 

Molecular weight: 463.5

CAS: 1261393-15-0

Purity: ≥99% deuterated forms (d1-d3)

Formulation: A solid

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Isotopically Labeled Standards|13C||Product Type|Biochemicals|Isotopically Labeled Standards|Deuterium||Product Type|Biochemicals|Small Molecule Inhibitors|MMPs||Product Type|Biochemicals|Small Molecule Inhibitors|Peptidases & Proteases||Research Area|Cardiovascular System|Blood|Coagulation & Hemostasis||Research Area|Cardiovascular System|Blood|Thrombosis

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