An inhibitor of HIV protease (Ki = 0.04 nM); inhibits the cytopathic effects of HIV-1 in MT-4 cells (IC50 = 150 nM)

Amprenavir – 25 mg

Brand:
Cayman
CAS:
161814-49-9
Storage:
-20
UN-No:
Non-Hazardous - /

Amprenavir is an inhibitor of HIV protease (Ki = 0.04 nM).{25257} It inhibits the cytopathic effects of HIV-1 in MT-4 cells (IC50 = 150 nM). Formulations containing amprenavir have been used in combination with other antiretroviral agents in the treatment of HIV-1 infection.  

 

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Description

An inhibitor of HIV protease (Ki = 0.04 nM); inhibits the cytopathic effects of HIV-1 in MT-4 cells (IC50 = 150 nM)

Formal name: N-[(1S,2R)-3-[[(4-aminophenyl)sulfonyl](2-methylpropyl)amino]-2-hydroxy-1-(phenylmethyl)propyl]-carbamic acid, (3S)-tetrahydro-3-furanyl ester

Synonyms:  141W94|APV|Prozei|VX-478

Molecular weight: 505.6

CAS: 161814-49-9

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Antivirals|Protease Inhibitors||Product Type|Biochemicals|Small Molecule Inhibitors|Peptidases & Proteases||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Viral Diseases|HIV & AIDS

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