A prodrug of piroxicam; converted to piroxicam at a rate of 100

Ampiroxicam – 500 mg

Brand:
Cayman
CAS:
99464-64-9
Storage:
-20
UN-No:
Non-Hazardous - /

Ampiroxicam is a prodrug of piroxicam (Item No. 13368), a non-steroidal anti-inflammatory drug (NSAID) that non-selectively and reversibly inhibits COX-1 and COX-2 (IC50s = 1.57 and 1.69 μM, respectively).{38295,17755} Ampiroxicam is converted to piroxicam at a rate of 100, 90, 70, and 50% in humans, rats, dogs, and monkeys, respectively.{38295}  

 

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SKU: 23026 - 500 mg Category:

Description

A prodrug of piroxicam; converted to piroxicam at a rate of 100, 90, 70, and 50% in humans, rats, dogs, and monkeys, respectively,

Formal name: carbonic acid, ethyl 1-[[2-methyl-1,1-dioxido-3-[(2-pyridinylamino)carbonyl]-2H-1,2-benzothiazin-4-yl]oxy]ethyl ester

Synonyms:  CP 65,703

Molecular weight: 447.5

CAS: 99464-64-9

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Cyclooxygenases||Research Area|Immunology & Inflammation|Arthritis (Non-autoimmune)||Research Area|Immunology & Inflammation|Inflammatory Lipid Mediators|Prostaglandins

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