An adamantoylindole derivative with an N-methylpiperidin-2-ylmethyl substitution at the indole 1-position that reportedly acts as a moderately potent agonist for both the CB1 and CB2 receptors (Kis = 11.9 and 4.8 nM

AM1248 – 5 mg

Brand:
Cayman
CAS:
335160-66-2
Storage:
-20
UN-No:
Non-Hazardous - /

AM1248 is an adamantoylindole derivative with an N-methylpiperidin-2-ylmethyl substitution at the indole 1-position. It reportedly acts as a moderately potent agonist for both the central CB1 and peripheral CB2 cannabinoid receptors (Kis = 11.9 and 4.8 nM, respectively).{20430} A related compound, 1-pentyl-3-(1-adamantoyl)indole, along with another synthetic cannabinoid, AM679, was identified as having been sold as a cannabinoid herbal blend known as “smart products” in Hungary in 2011.{20431}  

 

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Description

An adamantoylindole derivative with an N-methylpiperidin-2-ylmethyl substitution at the indole 1-position that reportedly acts as a moderately potent agonist for both the CB1 and CB2 receptors (Kis = 11.9 and 4.8 nM, respectively)

Formal name: [1-[(1-methyl-2-piperidinyl)methyl]-1H-indol-3-yl]tricyclo[3.3.1.13,7]dec-1-yl-methanone

Synonyms: 

Molecular weight: 390.6

CAS: 335160-66-2

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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