A synthetic progestin; an agonist of progesterone and androgen receptors (EC50s = 0.64 and 0.63 nM

Altrenogest – 1 g

Brand:
Cayman
CAS:
850-52-2
Storage:
-20
UN-No:
Non-Hazardous - /

Altrenogest is a synthetic progestin and an agonist of progesterone and androgen receptors (EC50s = 0.64 and 0.63 nM, respectively, in S. cerevisiae cells expressing human receptors).{40099} In vivo, altrenogest (20 mg/animal per day) reduces testicular weight, sperm content, and serum levels of luteinizing hormone and testosterone in boars.{47440} Altrenogest (0.044 mg/kg) increases serum concentrations of equine chorionic gonadotropin and embryonic size in pregnant mares.{47441} It also decreases genital perfusion and increases estrus cycle length in mares.{47442} Formulations containing altrenogest have been used to synchronize estrus in horses and pigs.  

 

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SKU: 27218 - 1 g Category:

Description

A synthetic progestin; an agonist of progesterone and androgen receptors (EC50s = 0.64 and 0.63 nM, respectively, in S. cerevisiae cells expressing human receptors); reduces testicular weight, sperm content, and serum levels of luteinizing hormone and testosterone in boars at 20 mg/animal per day; increases serum concentrations of equine chorionic gonadotropin and embryonic size in pregnant mares at 0.044 mg/kg; decreases genital perfusion and increases estrus cycle length in mares

Formal name: (17β)-17-hydroxy-17-(2-propen-1-yl)-estra-4,9,11-trien-3-one

Synonyms:  Allyltrenbolone|DRC 6246|RU 2267

Molecular weight: 310.4

CAS: 850-52-2

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Lipids|Sterol Lipids||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Androgens||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Estrogens & Progestins||Research Area|Endocrinology & Metabolism|Reproductive Biology

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