A synthetic CB which has a higher affinity for the peripheral CB2 receptor (Ki = 0.64 nM) over the central CB1 receptor (Ki = 270 nM); displays analgesic

A-836339 – 10 mg

Brand:
Cayman
CAS:
959746-77-1
Storage:
-20
UN-No:
Non-Hazardous - /

A-836339 is a synthetic cannabinoid (CB) which has a higher affinity for the peripheral CB2 receptor (Ki = 0.64 nM) over the central CB1 receptor (Ki = 270 nM).{21227} It displays analgesic, anti-inflammatory, and anti-hyperalgesic effects in mice.{21227}{23124} At higher doses, A-836339 also decreases spontaneous locomotor activities, consistent with CB1 activation.{21227} This product is intended for forensic and research applications.  

 

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Description

A synthetic CB which has a higher affinity for the peripheral CB2 receptor (Ki = 0.64 nM) over the central CB1 receptor (Ki = 270 nM); displays analgesic, anti-inflammatory, and anti-hyperalgesic effects in mice

Formal name: [N(Z)]-N-[3-(2-methoxyethyl)-4,5-dimethyl-2(3H)-thiazolylidene]-2,2,3,3-tetramethyl-cyclopropanecarboxamide

Synonyms: 

Molecular weight: 310.5

CAS: 959746-77-1

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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