A synthetic CB that shows high selectivity for the CB2 receptor (Ki = 0.77 nM) over the CB1 receptor (Ki = 2

A-796260 – 5 mg

Brand:
Cayman
CAS:
895155-26-7
Storage:
-20
UN-No:
Non-Hazardous - /

A-796260 is a synthetic cannabinoid (CB) that shows high selectivity for the CB2 receptor (Ki = 0.77 nM) over the CB1 receptor (Ki = 2,100 nM).{21031} It also shows efficacy in vivo in models of inflammatory, post-operative, neuropathic, and osteoarthritic pain, activities which are selectively blocked by CB2 receptor-selective antagonists.{21542} This product is intended for research and forensic uses.  

 

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SKU: 11606 - 5 mg Category:

Description

A synthetic CB that shows high selectivity for the CB2 receptor (Ki = 0.77 nM) over the CB1 receptor (Ki = 2,100 nM); shows efficacy in vivo in models of pain and is selectively blocked by CB2 receptor-selective antagonists; intended for research and forensic uses

Formal name: [1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl](2,2,3,3-tetramethylcyclopropyl)-methanone

Synonyms:  LTI-258

Molecular weight: 354.5

CAS: 895155-26-7

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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