An agonist at the µ-opioid receptor (pD2 = 8.20 µM)

7-hydroxy Mitragynine – 1 mg

Brand:
Cayman
CAS:
174418-82-7
Storage:
-20
UN-No:
Non-Hazardous - /

7-hydroxy Mitragynine (Item No. 13114) is an analytical reference standard that is structurally categorized as an opioid. It is an active metabolite of mitragynine (Item Nos. 18567 | 11151) that can be detected in urine.{33910} It is an agonist at the µ-opioid receptor (pD2 = 8.20), with a potency 13- and 46-fold higher than morphine and mitragynine, respectively.{20202} This product is intended for research and forensic applications.  

 

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Description

An agonist at the µ-opioid receptor (pD2 = 8.20 µM), with a potency 13- and 46-fold higher than mitragynine and morphine, respectively

Formal name: (αE,2S,3S,7aS,12bS)-3-ethyl-1,2,3,4,6,7,7a,12b-octahydro-7a-hydroxy-8-methoxy-α-(methoxymethylene)-indolo[2,3-a]quinolizine-2-acetic acid, methyl ester

Synonyms:  9-methoxy Corynantheidine Hydroxyindolenine

Molecular weight: 414.5

CAS: 174418-82-7

Purity: ≥98%

Formulation: A crystalline solid

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Opioids

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