A prodrug for methylprednisolone; has superior water solubility compared to the active glucocorticoid

6α-Methylprednisolone 21-hemisuccinate – 25 mg

Brand:
Cayman
CAS:
2921-57-5
Storage:
-20
UN-No:
Non-Hazardous - /

Methylprednisolone is a synthetic glucocorticoid that has anti-inflammatory and immunosuppressant effects through the glucocorticoid receptor.{19136} The methyl group reduces specific binding to corticosteroid-binding globulin, which may allow better tissue penetration, compared to that of prednisolone.{19136} 6α-Methylprednisolone 21-hemisuccinate is a prodrug for methylprednisolone.{21229} This compound has superior water solubility compared to the active glucocorticoid.{21228}  

 

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SKU: 11800 - 25 mg Category:

Description

A prodrug for methylprednisolone; has superior water solubility compared to the active glucocorticoid

Formal name: 21-(3-carboxy-1-oxopropoxy)-11β,17-dihydroxy-6α-methyl-pregna-1,4-diene-3,20-dione

Synonyms: 

Molecular weight: 474.6

CAS: 2921-57-5

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Receptor Pharmacology||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Glucocorticoids & Mineralocorticoids||Research Area|Immunology & Inflammation|Immunosuppressants

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