A pyridinium salt with anticholinesterase and antiproliferative activities; inhibits cholinesterase activity in rat brain homogenates (Kd = 33 μM); inhibits and yeast ChoK (IC50 = 17 μM); has antiproliferative activity against HT-29 colon cancer cells (IC50 = 2 μM)

4-(Dimethylamino)-1-methylpyridinium (iodide) – 50 mg

Brand:
Cayman
CAS:
7538-79-6
Storage:
-20
UN-No:
Non-Hazardous - /

4-(Dimethylamino)-1-methylpyridinium is a monoquaternary pyridinium salt with anticholinesterase and antiproliferative activities.{46209,46210} It inhibits cholinesterase activity in rat brain homogenates with a Kd value of 33 μM and yeast choline kinase (ChoK) with an IC50 value of 17 μM. 4-(Dimethylamino)-1-methylpyridinium also has antiproliferative activity against HT-29 colon cancer cells (IC50 = 2 μM).{46210}  

 

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SKU: 25861 - 50 mg Category:

Description

A pyridinium salt with anticholinesterase and antiproliferative activities; inhibits cholinesterase activity in rat brain homogenates (Kd = 33 μM); inhibits and yeast ChoK (IC50 = 17 μM); has antiproliferative activity against HT-29 colon cancer cells (IC50 = 2 μM)

Formal name: 4-(dimethylamino)-1-methyl-pyridinium, monoiodide

Synonyms: 

Molecular weight: 264.1

CAS: 7538-79-6

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Kinase Inhibitors||Product Type|Biochemicals|Small Molecule Inhibitors|Acetylcholine Turnover||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Cancer||Research Area|Neuroscience

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