An Mcl-1 inhibitor (Ki = 59 μM for binding of FITC-Mcl-1-BH2 peptide binding to Mcl-1); has been used as a building block in the synthesis of inhibitors of Mcl-1

3,6-dichloro-benzo[b]thiophene-2-Carboxylic Acid – 100 mg

Brand:
Cayman
CAS:
34576-94-8
Storage:
-20
UN-No:
Non-Hazardous - /

3,6-dichloro-benzo[b]thiophene-2-Carboxylic acid is an inhibitor of myeloid cell leukemia 1 (Mcl-1) with a Ki value of 59 μM for binding of FITC-Mcl-1-BH2 peptide binding to Mcl-1.{36227} It has been used as a building block in the synthesis of inhibitors of Mcl-1, the toll-like receptor 3/double-stranded RNA (TLR3/dsRNA) complex, and D-amino acid oxidase (DAO).{36227,36228,36229}  

 

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SKU: 22948 - 100 mg Category:

Description

An Mcl-1 inhibitor (Ki = 59 μM for binding of FITC-Mcl-1-BH2 peptide binding to Mcl-1); has been used as a building block in the synthesis of inhibitors of Mcl-1, the TLR3/dsRNA complex, and DAO

Formal name: 3,6-dichloro-benzo[b]thiophene-2-carboxylic acid

Synonyms: 

Molecular weight: 247.1

CAS: 34576-94-8

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors||Product Type|Biochemicals|Synthetic Intermediates & Building Blocks||Research Area|Cell Biology|Cell Death|Apoptosis

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