A triterpene with diverse biological activities; inhibits ADP-

3-Acetylursolic Acid – 5 mg

Brand:
Cayman
CAS:
7372-30-7
Storage:
-20
UN-No:
Non-Hazardous - /

3-Acetylursolic acid is a triterpene and derivative of ursolic acid (Item No. 10072) with diverse biological activities.{46903,46904,46905} It inhibits ADP-, thrombin-, or epinephrine-induced aggregation of isolated rat platelets (IC50s = P. falciparum in vitro (IC50 = 4 µM).{46904} It is also active against B. cereus, S. aureus, and S. pneumoniae (MICs = 39.1, 19.6, and 4.81 µM, respectively).{46905} It is cytotoxic to HepG2 cells (LC50 = 351 µM).  

 

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Description

A triterpene with diverse biological activities; inhibits ADP-, thrombin-, or epinephrine-induced aggregation of isolated rat platelets (IC50s = P. falciparum in vitro (IC50 = 4 µM); active against B. cereus, S. aureus, and S. pneumoniae (MICs = 39.1, 19.6, and 4.81 µM, respectively); cytotoxic to HepG2 cells (LC50 = 351 µM)

Formal name: 3β-(acetyloxy)-urs-12-en-28-oic acid

Synonyms:  Ursolic Acid Acetate

Molecular weight: 498.7

CAS: 7372-30-7

Purity: ≥95%

Formulation: A crystalline solid

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