A process-related impurity commonly found in the bulk synthesis of candesartan cilexetil

1H-1-ethyl Candesartan Cilexetil – 5 mg

Brand:
Cayman
CAS:
914613-35-7
Storage:
-20
UN-No:
Non-Hazardous - /

Candesartan cilexetil (Item No. 10489) is a prodrug of the potent, long-acting, and selective angiotensin II type 1 receptor (AT1) antagonist, candesartan. Clinical trials indicate a 4-16 mg/day dose of candesartan cilexetil effectively reduces diastolic blood pressure.{18425} 1H-1-ethyl Candesartan cilexetil is a process-related impurity commonly found in the bulk synthesis of candesartan cilexetil.{29093}  

 

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Description

A process-related impurity commonly found in the bulk synthesis of candesartan cilexetil

Formal name: 2-ethoxy-1-[[2′-(1-ethyl-1H-tetrazol-5-yl)[1,1′-biphenyl]-4-yl]methyl]-1H-benzimidazole-7-carboxylic acid, 1-[[(cyclohexyloxy)carbonyl]oxy]ethyl ester

Synonyms: 

Molecular weight: 638.7

CAS: 914613-35-7

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Pharmaceutical Impurities||Research Area|Cardiovascular System|Cardiovascular Diseases|Hypertension||Research Area|Neuroscience

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