A lipophilic analog of 17-phenyl trinor PGF2α

17-phenyl trinor Prostaglandin F2α methyl ester – 10 mg

Brand:
Cayman
CAS:
38315-47-8
Storage:
-20
UN-No:
Excepted Quantity - 1170 / 3

Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor. 17-phenyl trinor PGF2α methyl ester is a lipophilic analog of 17-phenyl trinor PGF2α, a potent agonist for the FP receptor. 17-phenyl trinor PGF2α binds the FP receptor on ovine luteal cells with a relative potency of 756% compared to that of PGF2α.{2058} Esters of PGs serve as prodrugs, as they are efficiently hydrolyzed in certain tissues to generate the bioactive free acid.  

 

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SKU: 10010110 - 10 mg Category:

Description

A lipophilic analog of 17-phenyl trinor PGF2α, a potent agonist for the FP receptor

Formal name: 7-[3R,5S-dihydroxy-2R-[3S-hydroxy-5Z-phenyl-1R-penten-1E-yl]cyclopentyl]-5-heptenoic acid, methyl ester

Synonyms:  17-phenyl trinor PGF2α methyl ester|Bimatoprost methyl ester

Molecular weight: 402.5

CAS: 38315-47-8

Purity: ≥98%

Formulation: A solution in ethanol

Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Receptor Pharmacology|Agonists||Research Area|Endocrinology & Metabolism|Reproductive Biology||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway||Research Area|Neuroscience|Ophthalmology

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