15(R)-PGE1 is the “unnatural” C-15 stereoisomer of PGE1. It is essentially inactive biologically when compared to PGE1.{1350} It is a non-competitive inhibitor of 15-hydroxy PGDH with an IC50 of 189 µM.{2274}

15(R)-Prostaglandin E1 – 5 mg

Brand:
Cayman
CAS:
20897-91-0
Storage:
-20
UN-No:
De Minimis - 1231 / 3

15(R)-PGE1 is the “unnatural” C-15 stereoisomer of PGE1. It is essentially inactive biologically when compared to PGE1.{1350} It is a non-competitive inhibitor of 15-hydroxy PGDH with an IC50 of 189 µM.{2274}  

 

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Description

15(R)-PGE1 is the “unnatural” C-15 stereoisomer of PGE1. It is essentially inactive biologically when compared to PGE1.{1350} It is a non-competitive inhibitor of 15-hydroxy PGDH with an IC50 of 189 µM.{2274}

Formal name: 9-oxo-11α,15R-dihydroxy-prost-13E-en-1-oic acid

Synonyms:  15(R)-PGE1|15-epi PGE1

Molecular weight: 354.5

CAS: 20897-91-0

Purity: ≥95%

Formulation: A solution in methyl acetate

Product Type|Biochemicals|Lipids|Prostaglandins||Product Type|Biochemicals|Small Molecule Inhibitors||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway

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