An epimer of PTA2; does not inhibit collagen-induced platelet aggregation (IC50s = 120-130 µM); does not affect gastric tone in isolated rat gastric fundus when used at concentrations of 0.5 or 1.5 µg/ml; less effective than PTA2 at inhibiting prostaglandin-induced contraction of isolated rat stomach muscle

15(R)-Pinane Thromboxane A2 – 1 mg

Brand:
Cayman
CAS:
71154-83-1
Storage:
-20
UN-No:
De Minimis - 1170 / 3

15(R)-Pinane thromboxane A2 is the (R)-epimer of pinane thromboxane A2 (PTA2; Item No. 19020). 15(R)-PTA2 does not inhibit collagen-induced platelet aggregation (IC50s = 120-130 µM).{41363} It does not affect gastric tone in isolated rat gastric fundus when used at concentrations of 0.5 or 1.5 µg/ml and is less effective than PTA2 at inhibiting prostaglandin-induced contraction of isolated rat stomach muscle.{41364}  

 

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SKU: 10008510 - 1 mg Category:

Description

An epimer of PTA2; does not inhibit collagen-induced platelet aggregation (IC50s = 120-130 µM); does not affect gastric tone in isolated rat gastric fundus when used at concentrations of 0.5 or 1.5 µg/ml; less effective than PTA2 at inhibiting prostaglandin-induced contraction of isolated rat stomach muscle

Formal name: (5Z)-7-[(1S,2R,3R,5S)-3-[(1E,3R)-3-hydroxy-1-octen-1-yl]-6,6-dimethylbicyclo[3.1.1]hept-2-yl]-5-heptenoic acid

Synonyms:  15(R)-PTA2|15-epi-Pinane Thromboxane A2|15-epi-PTA2|15-iso-Pinane Thromboxane A2|15-iso-PTA2

Molecular weight: 376.6

CAS: 71154-83-1

Purity: >98%

Formulation: A solution in ethanol

Product Type|Biochemicals|Lipids|Thromboxanes||Research Area|Cardiovascular System||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway

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