11β-PGE2 is the C-11 epimer of PGE2. It is a moderate inhibitor of PGE2 binding to rat hypothalamic membranes with a Ki value of 53 nM.{1924} 11β-PGE2 also stimulates bone resorption in rats at concentrations of 10-8 to 10-6 M which is similar to PGE2.{2052} 11β-PGE2 inhibits PGE2 binding to the prostaglandin transporter protein with a Ki of 56 nM.{3806}

11β-Prostaglandin E2 – 1 mg

Brand:
Cayman
CAS:
38310-90-6
Storage:
-20
UN-No:
De Minimis - 1231 / 3

11β-PGE2 is the C-11 epimer of PGE2. It is a moderate inhibitor of PGE2 binding to rat hypothalamic membranes with a Ki value of 53 nM.{1924} 11β-PGE2 also stimulates bone resorption in rats at concentrations of 10-8 to 10-6 M which is similar to PGE2.{2052} 11β-PGE2 inhibits PGE2 binding to the prostaglandin transporter protein with a Ki of 56 nM.{3806}  

 

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Description

11β-PGE2 is the C-11 epimer of PGE2. It is a moderate inhibitor of PGE2 binding to rat hypothalamic membranes with a Ki value of 53 nM.{1924} 11β-PGE2 also stimulates bone resorption in rats at concentrations of 10-8 to 10-6 M which is similar to PGE2.{2052} 11β-PGE2 inhibits PGE2 binding to the prostaglandin transporter protein with a Ki of 56 nM.{3806}

Formal name: 9-oxo-11β,15S-dihydroxy-prosta-5Z,13E-dien-1-oic acid

Synonyms:  11-epi PGE2|11β-PGE2

Molecular weight: 352.5

CAS: 38310-90-6

Purity: ≥98%

Formulation: A solution in methyl acetate

Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Endocrinology & Metabolism|Bone Growth & Remodeling||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway

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