An internal standard for the quantification of (±)-JWH 018 N-(4-hydroxypentyl) metabolite by GC- or LC-MS

(±)-JWH 018 N-(4-hydroxypentyl) metabolite-d5 – 500 µg

Brand:
Cayman
CAS:
1413427-49-2
Storage:
-20
UN-No:
De Minimis - 1230 / 3|6.1

(±)-JWH 018 N-(4-hydroxypentyl) metabolite-d5 contains five deuterium atoms at the 2, 5, 6, 7, and 8 positions. It is intended for use as an internal standard for the quantification of (±)-JWH 018 N-(4-hydroxypentyl) metabolite by GC- or LC-mass spectrometry. JWH 018 is a mildly selective agonist of the peripheral cannabinoid (CB2) receptor, derived from the aminoalkylindole WIN 55,212-2. The Ki values for binding central cannabinoid (CB1) and CB2 receptors are 9.0 and 2.94 nM, respectively, for a CB1:CB2 ratio of 3.06.{16797} JWH 018 is one of several synthetic CBs which have been included in smoking mixtures.{18291,19507} (±)-JWH 018 N-(4-hydroxypentyl) metabolite is a urinary metabolite of JWH 018, characterized by monohydroxylation of the N-alkyl chain.{19353} Its biological actions are unknown.  

 

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SKU: 10926 - 500 µg Category:

Description

An internal standard for the quantification of (±)-JWH 018 N-(4-hydroxypentyl) metabolite by GC- or LC-MS

Formal name: (1-(4-hydroxypentyl)-2,5,6,7,8-d5-1H-indol-3-yl)(naphthalen-1-yl)-methanone

Synonyms: 

Molecular weight: 362.5

CAS: 1413427-49-2

Purity: ≥99% deuterated forms (d1-d5)

Formulation: A solution in methanol

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Drugs of Abuse||Product Type|Biochemicals|Isotopically Labeled Standards|Deuterium||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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