A bicyclic CB analog that avidly binds the CB1 receptor (Ki = 0.83 nM) and shows high antinociceptive activity; ten-fold more potent than Δ9-THC in analgesic

(±)-CP 47,497-C8-homolog (exempt preparation) – 5 mg

Brand:
Cayman
CAS:
70434-92-3
Storage:
-20
UN-No:
De Minimis - 1230 / 3|6.1

(±)-CP 47,497-C8-homolog is a bicyclic cannabinoid (CB) analog that avidly binds the CB1 receptor (Ki = 0.83 nM) and shows high antinociceptive activity.{6746} It is ten-fold more potent than Δ9-tetrahydrocannabinol in analgesic, motor depressant, anticonvulsant, and hypothermic effects in mice.{17059}  

 

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Description

A bicyclic CB analog that avidly binds the CB1 receptor (Ki = 0.83 nM) and shows high antinociceptive activity; ten-fold more potent than Δ9-THC in analgesic, motor depressant, anticonvulsant, and hypothermic effects in mice

Formal name: rel-2-[(1S,3R)-3-hydroxycyclohexyl]-5-(2-methylnonan-2-yl)phenol

Synonyms:  Cannabicyclohexanol|CAY10596

Molecular weight: 332.5

CAS: 70434-92-3

Purity: ≥98%

Formulation: A solution in methanol

Product Type|Biochemicals|Drugs of Abuse||Research Area|Forensic Chemistry & Toxicology|Cannabinoids|Synthetic Cannabinoids

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