(±)-Cloprostenol (sodium salt) is a more water solute

(±)-Cloprostenol (sodium salt) – 1 mg

Brand:
Cayman
CAS:
55028-72-3
Storage:
-20
UN-No:
Non-Hazardous - /

(±)-Cloprostenol (sodium salt) is a more water solute, crystalline form of cloprostenol than the free acid. Cloprostenol is a synthetic analog of prostaglandin F2α (PGF2α; Item No. 16010). It is 200 times and 100 times more potent than PGF2α in terminating pregnancy in hamsters and rats, respectively, without the side effects associated with PGF2α.{1182} The subcutaneous dose required for interrupting early pregnancy is species dependent, requiring approximately 1.25 µg/kg and 270 µg/kg in hamsters and rats, respectively.{1182} Cloprostenol is also a potent inhibitor of rat adipose precursor differentiation in primary cultures with an IC50 of 3 x 10−12 M.{4404}  

 

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Description

(±)-Cloprostenol (sodium salt) is a more water solute, crystalline form of cloprostenol than the free acid.

Formal name: (±)-9α,11α,15R-trihydroxy-16-(3-chlorophenoxy)-17,18,19,20-tetranor-prosta-5Z,13E-dien-1-oic acid, sodium salt

Synonyms:  (±)-16-m-chlorophenoxy tetranor PGF2α|(±)-16-m-chlorophenoxy tetranor Prostaglandin F2α|DL-Cloprostenol

Molecular weight: 446.9

CAS: 55028-72-3

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Lipids|Prostaglandins||Research Area|Endocrinology & Metabolism|Reproductive Biology||Research Area|Lipid Biochemistry|Cyclooxygenase Pathway

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