A bioactive metabolite of amphetamine that acts as an agonist of the trace amine-associated receptor 1 (EC50 = ~0.2 μM in HEK293 cells expressing rat TAAR1); used to dilate the pupil in the diagnosis of Horner’s syndrome; intended only for forensic and research purposes

4-hydroxy Amphetamine (hydrochloride) – 10 mg

Brand:
Cayman
CAS:
876-26-6
Storage:
-20
UN-No:
Non-Hazardous - /

4-Hydroxyamphetamine (4-HA) is a bioactive metabolite of amphetamine.{24225,24227} This sympathomimetic is an agonist of the trace amine-associated receptor 1 (EC50 = ~0.2 μM in HEK293 cells expressing rat TAAR1).{24228} As a 1% ophthalmologic solution, 4-HA has been used to dilate the pupil in the diagnosis of Horner’s syndrome.{24224,24226} This product is intended only for forensic and research purposes.  

 

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SKU: 9001830 - 10 mg Category:

Description

A bioactive metabolite of amphetamine that acts as an agonist of the trace amine-associated receptor 1 (EC50 = ~0.2 μM in HEK293 cells expressing rat TAAR1); used to dilate the pupil in the diagnosis of Horner’s syndrome; intended only for forensic and research purposes

Formal name: 4-​(2-​aminopropyl)​-phenol, monohydrochloride

Synonyms:  p-hydroxy Amphetamine|para-hydroxy Amphetamine|4-HA|Paredrine|POHA|α-methyl Tyramine

Molecular weight: 187.7

CAS: 876-26-6

Purity: ≥98%

Formulation: A crystalline solid

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