An antitubercular agent; active against clinical isolates of drug-resistant and -sensitive replicating M. tuberculosis (MICs = M. tuberculosis over M. scrofulaceum

TBA-354 – 100 mg

Brand:
Cayman
CAS:
1257426-19-9
Storage:
-20
UN-No:
Non-Hazardous - /

TBA-354 is a nitroimidazole antitubercular agent.{46935} It is active against clinical isolates of drug-resistant and -sensitive replicating M. tuberculosis (MICs = M. tuberculosis over M. scrofulaceum, M. gilvum, M. fortuitum, M. triviale, and M. smegmatis (MICs = >11.5 μM) but is active against M. bovis and M. kansasii (MICs = M. tuberculosis infection.  

 

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SKU: 30317 - 100 mg Category:

Description

An antitubercular agent; active against clinical isolates of drug-resistant and -sensitive replicating M. tuberculosis (MICs = M. tuberculosis over M. scrofulaceum, M. gilvum, M. fortuitum, M. triviale, and M. smegmatis (MICs = >11.5 μM) but is active against M. bovis and M. kansasii (MICs = M. tuberculosis infection at 100 mg/kg per day

Formal name: (6S)-6,7-dihydro-2-nitro-6-[[6-[4-(trifluoromethoxy)phenyl]-3-pyridinyl]methoxy]-5H-imidazo[2,1-b][1,3]oxazine

Synonyms: 

Molecular weight: 436.3

CAS: 1257426-19-9

Purity: ≥98%

Formulation: A crystalline solid

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