An active metabolite of ivabradine

N-desmethyl Ivabradine (hydrochloride) – 5 mg

Brand:
Cayman
CAS:
1246638-08-3
Storage:
-20
UN-No:
De Minimis - 3077 / 9

N-desmethyl Ivabradine is an active metabolite of ivabradine (Item No. 15868).{42971} Ivabradine is metabolized by the cytochrome P450 (CYP) isoform CYP3A4.  

 

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SKU: 27808 - 5 mg Category:

Description

An active metabolite of ivabradine

Formal name: 3-[3-[[[(7S)-3,4-dimethoxybicyclo[4.2.0]octa-1,3,5-trien-7-yl]methyl]amino]propyl]-1,3,4,5-tetrahydro-7,8-dimethoxy-2H-3-benzazepin-2-one, monohydrochloride

Synonyms: 

Molecular weight: 491

CAS: 1246638-08-3

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Ion Channel Modulation|Blockers||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Cardiovascular System|Cardiovascular Diseases|Angina||Research Area|Cardiovascular System|Cardiovascular Diseases|Heart Failure||Research Area|Cardiovascular System|Cardiovascular Diseases|Myocardial Infarction||Research Area|Cardiovascular System|Heart|Arrhythmia||Research Area|Toxicology|Drug Metabolism|Drug Metabolites

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