An inactive metabolite of abacavir; formed from abacavir via reactive aldehyde intermediates that can form adducts with proteins

Abacavir Carboxylate – 1 mg

Brand:
Cayman
CAS:
384380-52-3
Storage:
-20
UN-No:
Non-Hazardous - /

Abacavir carboxylate is an inactive metabolite of the HIV-1 reverse transcriptase inhibitor abacavir (Item No. 14746).{43845,43846} It is formed from abacavir via reactive aldehyde intermediates that can form adducts with proteins on valine residues.{43846}  

 

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SKU: 27777 - 1 mg Category:

Description

An inactive metabolite of abacavir; formed from abacavir via reactive aldehyde intermediates that can form adducts with proteins

Formal name: (1S,4R)-4-[2-amino-6-(cyclopropylamino)-9H-purin-9-yl]-2-cyclopentene-1-carboxylic acid

Synonyms: 

Molecular weight: 300.3

CAS: 384380-52-3

Purity: ≥95%

Formulation: A solid

Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Viral Diseases|HIV & AIDS||Research Area|Toxicology|Drug Metabolism|Drug Metabolites

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