An antimalarial compound; inhibits recombinant P. vivax and human PI4K (IC50s = 3.5 and 90 nM

BQR-695 – 10 mg

Brand:
Cayman
CAS:
1513879-21-4
Storage:
-20
UN-No:
Non-Hazardous - /

BQR-695 is an antimalarial compound.{53056} It inhibits recombinant P. vivax and human phosphatidylinositol 4-kinase (PI4K; IC50s = 3.5 and 90 nM, respectively). BQR-695 induces schizont-stage arrest and death of P. falciparum (IC50 = ~70 nM) without inducing cytotoxicity in mature red blood cells (RBCs).  

 

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SKU: 27482 - 10 mg Category:

Description

An antimalarial compound; inhibits recombinant P. vivax and human PI4K (IC50s = 3.5 and 90 nM, respectively); induces schizont-stage arrest and death of P. falciparum (IC50 = ~70 nM)

Formal name: 2-[[7-(3,4-dimethoxyphenyl)-2-quinoxalinyl]amino]-N-methyl-acetamide

Synonyms: 

Molecular weight: 352.4

CAS: 1513879-21-4

Purity: ≥98%

Formulation: A solid

Product Type|Biochemicals|Antiparasitics|Antiprotozoals||Product Type|Biochemicals|Kinase Inhibitors|Other Lipid Kinases||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Parasitic Diseases|Malaria

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