A metabolite of atazanavir

Des(benzylpyridyl) Atazanavir – 25 mg

Brand:
Cayman
CAS:
1192224-24-0
Storage:
-20
UN-No:
Non-Hazardous - /

Des(benzylpyridyl) atazanavir is a major metabolite of the HIV-1 protease inhibitor atazanavir (Item No. 11733).{46499,46500} It is formed from atazanavir by the cytochrome P450 (CYP) isoforms CYP3A4 and CYP2D6.{46500}  

 

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SKU: 27372 - 25 mg Category:

Description

A metabolite of atazanavir

Formal name: (3S,8S,9S,12S)-3,12-bis(1,1-dimethylethyl)-8-hydroxy-4,11-dioxo-9-(phenylmethyl)-2,5,6,10,13-pentaazatetradecanedioic acid 1,14-dimethyl ester

Synonyms:  Atazanavir metabolite M1

Molecular weight: 537.7

CAS: 1192224-24-0

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Antivirals|Protease Inhibitors||Product Type|Biochemicals|Small Molecule Inhibitors|Peptidases & Proteases||Product Type|Biochemicals|Xenobiotic Metabolites||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Viral Diseases|HIV & AIDS||Research Area|Toxicology|Drug Metabolism|Cytochrome P450||Research Area|Toxicology|Drug Metabolism|Drug Metabolites

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