An inhibitor of Glut1 (Ki = 15 µM); an inhibitor of the interaction between HIV-1 integrase and LEDGF/p75 (IC50 = 94.07 µM); a weak inhibitor of tyrosine kinases (IC50 = 0.49 µg/ml); and has been used as a negative control for lavendustin A

Lavendustin B – 5 mg

Brand:
Cayman
CAS:
125697-91-8
Storage:
-20
UN-No:
Non-Hazardous - /

Lavendustin B is a competitive inhibitor of glucose transporter 1 (Glut1; Ki = 15 µM).{46352} It is also an inhibitor of the interaction between HIV-1 integrase and LEDGF/p75 (IC50 = 94.07 µM).{46353} Lavendustin B is a weak inhibitor of tyrosine kinases (IC50 = 0.49 µg/ml) and has been used as a negative control for the protein tyrosine kinase inhibitor lavendustin A (Item No. 10010268).{16076,46354,46355}  

 

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SKU: 27311 - 5 mg Category:

Description

An inhibitor of Glut1 (Ki = 15 µM); an inhibitor of the interaction between HIV-1 integrase and LEDGF/p75 (IC50 = 94.07 µM); a weak inhibitor of tyrosine kinases (IC50 = 0.49 µg/ml); and has been used as a negative control for lavendustin A

Formal name: 5-[bis[(2-hydroxyphenyl)methyl]amino]-2-hydroxy-benzoic acid

Synonyms: 

Molecular weight: 365.4

CAS: 125697-91-8

Purity: ≥95%

Formulation: A crystalline solid

Product Type|Biochemicals|Ion Channel Modulation|Blockers||Product Type|Biochemicals|Kinase Inhibitors|EGFR/ErbB/HER Family||Product Type|Biochemicals|Small Molecule Inhibitors|Kinases||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Viral Diseases|HIV & AIDS||Research Area|Neuroscience

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