A PAD3 inhibitor (kinact/KI = 15

CAY10727 – 250 µg

Brand:
Cayman
CAS:
1671088-84-8
Storage:
-20
UN-No:
De Minimis - 1170 / 3

CAY10727 is an inhibitor of protein arginine deiminase 3 (PAD3; kinact/KI = 15,600 M-1min-1).{48907} It is selective for PAD3 over PAD1, -2, and -4 (kinact/KIs = 360, 1,110, and 1,460 M-1min-1, respectively).  

 

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SKU: 26543 - 250 µg Category:

Description

A PAD3 inhibitor (kinact/KI = 15,600 M-1min-1); selective for PAD3 over PAD1, -2, and -4 (kinact/KIs = 360, 1,110, and 1,460 M-1min-1, respectively)

Formal name: 2-chloro-N-[3-[1-[(2′-chloro[1,1′-biphenyl]-3-yl)methyl]-2,5-dioxo-4-imidazolidinyl]propyl]-ethanimidamide

Synonyms: 

Molecular weight: 433.3

CAS: 1671088-84-8

Purity: ≥90%

Formulation: A solution in ethanol

Product Type|Biochemicals|Small Molecule Inhibitors|Deiminases||Research Area|Epigenetics, Transcription, & Translation|Writers|Citrullination

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