A GABAA receptor ligand; accelerates decay of GABA-induced currents in HEK293 cells expressing rat α1β2

U-93631 – 10 mg

Brand:
Cayman
CAS:
152273-12-6
Storage:
-20
UN-No:
Non-Hazardous - /

U-93631 is a GABAA receptor ligand.{47207} It accelerates decay of GABA-induced currents in HEK293 cells expressing rat α1β2, β2γ2, and α1γ2 subunit-containing GABAA receptors when used at a concentration of 5 μM. U-93631 inhibits radioligand binding to the picrotoxin site on α1β2γ2 subunit-containing GABAA receptors.{47208}  

 

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SKU: 26417 - 10 mg Category:

Description

A GABAA receptor ligand; accelerates decay of GABA-induced currents in HEK293 cells expressing rat α1β2, β2γ2, and α1γ2 subunit-containing GABAA receptors at 5 μM; inhibits radioligand binding to the picrotoxin site on α1β2γ2 subunit-containing GABAA receptors

Formal name: 4,5-dihydro-4,4-dimethyl-imidazo[1,5-a]quinoxaline-3-carboxylic acid, 1,1-dimethylethyl ester

Synonyms: 

Molecular weight: 299.4

CAS: 152273-12-6

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Ion Channel Modulation||Research Area|Neuroscience

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