A VHL Ligand 1 derivative; comprises the VHL ligand domain and PEG linker of the BET inhibitor-containing PROTACs MZ2 and MZP-55

VH 032 Linker 2 – 50 mg

Brand:
Cayman
CAS:
2064292-52-8
Storage:
-20
UN-No:
Non-Hazardous - /

VH 032 Linker 2 is a derivative of the proteolysis-targeting chimera technology (PROTAC) building block VHL ligand 1 (Item No. 21591). VH 032 Linker 2 comprises the von Hippel-Lindau (VHL) ligand domain and the polyethylene glycol (PEG) linker of the bromodomain and extra terminal (BET) inhibitor-containing PROTACs MZ2 and MZP-55.{43633}  

 

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SKU: 26149 - 50 mg Category:

Description

A VHL Ligand 1 derivative; comprises the VHL ligand domain and PEG linker of the BET inhibitor-containing PROTACs MZ2 and MZP-55

Formal name: (2S,4R)-1-((S)-17-amino-2-(tert-butyl)-4-oxo-6,9,12,15-tetraoxa-3-azaheptadecanoyl)-4-hydroxy-N-(4-(4-methylthiazol-5-yl)benzyl)pyrrolidine-2-carboxamide, monohydrochloride

Synonyms:  E3 Ligase Ligand-Linker Conjugate 7

Molecular weight: 700.3

CAS: 2064292-52-8

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|PROTACs||Product Type|Biochemicals|Synthetic Intermediates & Building Blocks||Research Area|Cell Biology|Proteolysis|Ubiquitin/Proteasome System||Research Area|Epigenetics, Transcription, & Translation|Readers|Bromodomains

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