An internal standard for the quantification of varenicline by GC- or LC-MS

Varenicline-d4 – 1 mg

Brand:
Cayman
CAS:
2183239-01-0
Storage:
-20
UN-No:
Non-Hazardous - /

Varenicline-d4 is intended for use as an internal standard for the quantification of varenicline (Item No. 15030) by GC- or LC-MS. Varenicline is a full agonist of α7 subunit-containing neuronal nicotinic acetylcholine receptors (nAChRs; EC50 = 18 µM) and a partial agonist of α4β2 subunit-containing nAChRs (EC50 = 2.3 µM).{22776} Formulations containing varenicline have been used as aids in smoking cessation.  

 

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SKU: 26102 - 1 mg Category:

Description

An internal standard for the quantification of varenicline by GC- or LC-MS

Formal name: 7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g]quinoxaline-7,7,9,9-d4

Synonyms: 

Molecular weight: 215.3

CAS: 2183239-01-0

Purity: ≥99% deuterated forms (d1-d4)

Formulation: A solid

Application|Mass Spectrometry||Product Type|Biochemicals|Analytical Standards||Product Type|Biochemicals|Ion Channel Modulation|Activators||Product Type|Biochemicals|Isotopically Labeled Standards|Deuterium||Research Area|Neuroscience|Behavioral Neuroscience|Addiction Research

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