An isomer of KT109; a less potent inhibitor of DAGLβ (IC50 = 39.81 nM)

(S)-KT109 – 1 mg

Brand:
Cayman
CAS:
2055172-61-5
Storage:
-20
UN-No:
Non-Hazardous - /

(S)-KT109 is the (S) isomer of the diacylglycerol lipase β (DAGLβ) inhibitor KT109 (Item No. 18933).{43435} (S)-KT109 is a less potent inhibitor of DAGLβ (IC50 = 39.81 nM), DAGLα-mediated hydrolysis of 1-stearoyl-2-arachidonoyl-sn-glycerol (IC50 = 794.3 nM), and α/β-hydrolase domain-containing protein 6 (ABHD6; IC50 = 630.9 nM) than (R)-KT109 (Item No. 25682).  

 

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SKU: 25683 - 1 mg Category:

Description

An isomer of KT109; a less potent inhibitor of DAGLβ (IC50 = 39.81 nM), DAGLα-mediated hydrolysis of 1-stearoyl-2-arachidonoyl-sn-glycerol (IC50 = 794.3 nM), and ABHD6 (IC50 = 630.9 nM) than (R)-KT109

Formal name: (4-[1,1′-biphenyl]-4-yl-1H-1,2,3-triazol-1-yl)[(2S)-2-(phenylmethyl)-1-piperidinyl]-methanone

Synonyms: 

Molecular weight: 422.5

CAS: 2055172-61-5

Purity: ≥98%

Formulation: A crystalline solid

Product Type|Biochemicals|Small Molecule Inhibitors|Glycerolipid Lipases||Research Area|Lipid Biochemistry|Endocannabinoid/Endocannabinoid-like||Research Area|Lipid Biochemistry|Glycerolipids|Lipases||Research Area|Neuroscience

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