Description
An inhibitor of LDHA (Kd = 0.093 μM; IC50 = 0.5 μM); selective for LDHA over LDHB in an NADH competition assay using recombinant enzymes (IC50s = 0.54 and 3.6 μM, respectively); cell-impermeable and lacks cytotoxicity against HeLa cervical cancer cells (IC50 = >500 μM),
Formal name: 2-[[4-[4-[[3-[(2-methyl-6-benzothiazolyl)amino]-3-oxopropyl]amino]-4-oxobutyl]phenyl]methyl]-propanedioic acid
Synonyms:
Molecular weight: 497.6
CAS: 1370290-34-8
Purity: ≥98%
Formulation: A crystalline solid
Product Type|Biochemicals|Small Molecule Inhibitors||Research Area
