An inhibitor of N-myristoyltransferase (IC50 = 50 = >1

IMP-1088 – 10 mg

Brand:
Cayman
CAS:
2059148-82-0
Storage:
-20
UN-No:
Excepted Quantity - 1231 / 3

IMP-1088 is an inhibitor of N-myristoyltransferase 1 (NMT1) and NMT2 (IC50 = 50 = >1,000 nM). It also blocks production of infectious RV-16 virus in primary human bronchial epithelial cells (hBECs) when added 3 hours post infection via inhibition of viral capsid assembly.  

 

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SKU: 25366 - 10 mg Category:

Description

An inhibitor of N-myristoyltransferase (IC50 = 50 = >1,000 nM); blocks production of infectious RV-16 virus in primary hBECs

Formal name: 5-[3,4-difluoro-2-[2-(1,3,5-trimethyl-1H-pyrazol-4-yl)ethoxy]phenyl]-N,N,1-trimethyl-1H-indazole-3-methanamine

Synonyms: 

Molecular weight: 453.5

CAS: 2059148-82-0

Purity: ≥98%

Formulation: A solution in methyl acetate

Product Type|Biochemicals|Antivirals||Product Type|Biochemicals|Small Molecule Inhibitors|Acyltransferases||Research Area|Immunology & Inflammation||Research Area|Infectious Disease|Viral Diseases|Rhinoviruses

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