A synthetic progestogen; inhibits ovulation and prevents fertilization in rabbits and mice; inhibits rhodamine123 efflux

Desogestrel – 10 mg

Brand:
Cayman
CAS:
54024-22-5
Storage:
-20
UN-No:
De Minimis - 3077 / 9

Desogestrel is a synthetic progestogen.{41180} It inhibits ovulation and prevents fertilization in rabbits and mice. Desogestrel inhibits rhodamine123 efflux, a measure of P-glycoprotein activity, ex vivo in human lymphocytes and CD8+ T cells in a dose-dependent manner.{41181} Formulations containing desogestrel have been used as oral contraceptives and for the treatment of polycystic ovary syndrome.{41181,41182}  

 

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SKU: 23651 - 10 mg Category:

Description

A synthetic progestogen; inhibits ovulation and prevents fertilization in rabbits and mice; inhibits rhodamine123 efflux, a measure of P-glycoprotein activity, ex vivo in human lymphocytes and CD8+ T cells in a dose-dependent manner

Formal name: (17α)-13-ethyl-11-methylene-18,19-dinorpregn-4-en-20-yn-17-ol

Synonyms:  ORG 2969

Molecular weight: 310.5

CAS: 54024-22-5

Purity: ≥95%

Formulation: A solid

Product Type|Biochemicals|Lipids|Sterol Lipids||Product Type|Biochemicals|Transporter & Exchanger Modulators||Research Area|Endocrinology & Metabolism|Hormones & Receptors|Estrogens & Progestins||Research Area|Endocrinology & Metabolism|Reproductive Biology||Research Area|Toxicology|Drug Metabolism

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